I-CAS 112809-51-5 I-Anti Estrogen Steroid Powder White Henlthy Letrozole Femara Yomdlavuza Webele
Imininingwane Esheshayo
I-CAS: 112809-51-5
Synonimes:FEMARA;CGS-20267;LETROZOL;LETROZOLE;LetrozoleUsp28;Letrozole99%;CGS-20267, Femara
Ubumsulwa: 99%
Ukubukeka: Ikristalu emhlophe noma ekhanyayo ephuzi
I-Molecular Formula: C17H11N5
Isisindo se-molecule: 285.31
Indawo Encibilikayo: 181°C~183°C
I-Anti Estrogen Bodybuilding Steroids Letrozole Femara White Powder CAS 112809-51-5
Ukusetshenziswa: Kusetshenziswa njenge-API ekwelapheni isifo sebele.
Umthamo onconyiwe we-Femara yithebhulethi eyodwa engu-2.5 mg kanye ngosuku, ngaphandle kokubheka ukudla.
I-Letrozole yehlisa amazinga e-estrogen kwabesifazane abadlule kokuya esikhathini, okungase kubambezele ukukhula kwezinhlobo ezithile zezimila zamabele ezidinga i-estrogen ukuze zikhule emzimbeni.
Iresiphi ye-Letrozole
umthamo | impahla |
1 igramu | I-Letrozole powder |
19.9 ml | I-PEG 300 |
179.1 ml | 190 Ubufakazi Bezinhlamvu Zotshwala |
I-Letrozole/Femara Dosing
Abasebenzisi be-anecdotally baye babika ukuthi babone imiphumela emihle besebenzisa imithamo esukela cishe ku-.25mgs ngosuku ukuya ku-.5mgs ngosuku.Kodwa-ke le mithamo iyahluka kakhulu ukusuka kumsebenzisi kuye kumsebenzisi, okuhlanganisa namashejuli womthamo.Abanye baye babika ukusebenzisa i-compound njalo ngemva kwezinsuku ezintathu noma zonke izinsuku ezintathu ngemiphumela emihle.Futhi, amanani abikiwe asuka ku-.25mgs kuya ku-2.5mgs ngosuku.
Mayelana nomthamo, udinga ukukhetha ngokuhambisana nesimo somzimba wakho, noma uthintane nomqeqeshi/udokotela wakho.Le ndatshana ingeyereferensi kuphela.
I-Letrozole/Femara Effect
I-Letrozole ezigulini ze-postmenopausal ezinomdlavuza webele othuthukisiwe one-Estrogen receptor kanye / noma i-progesterone receptor positive noma isimo se-receptor esingaziwa
I-Femara (i-letrozole) iwuhlobo lwe-II (non-steroidal) lwesizukulwane sesithathu se-aromatase inhibitor.Ngokomtholampilo isetshenziselwa ukwelapha abesifazane abangemva kokuya esikhathini abane-estrogen receptor positive noma i-estrogen receptor engaziwa umdlavuza webele.
1. I-Letrozole iyi-Aromatase Inhibitor enamandla eyakhiwe ukulwa nomdlavuza webele.
2. Kwabagijimi nabakhi bomzimba, kuyisidakamizwa esisetshenziselwa ukulwa nemiphumela emibi ye-estrogenic ye-anabolic steroids ukugcinwa kwamanzi, induna kanye ne-gynocomastia.
3. Izophinde inyuse amazinga e-testosterone ngenxa yokwehla kwe-estrogen emzimbeni.
4. I-Femara(igama elijwayelekile lithi letrozole) umuthi omusha owenzelwe ukwelapha umdlavuza webele othuthukile kwabesifazane.
5. I-Femara ingeyesibili ekilasini elisha lama-oral aromatase inhibitors akhethiwe esizukulwaneni sesithathu.
6. Isebenza ngokuvimbela i-enzyme aromatase, kamuva ivimbele ukukhiqizwa kwe-estrogen.
Incazelo ye-Letrozole/Femara
Esihlokweni esisodwa sokuhlolwa kwabesilisa i-Letrozole yakwazi ukunciphisa amazinga e-estrogen kumazinga angabonakali.I-Letrozole iyakwazi ukukhulisa i-testosterone ezifundweni zesilisa.
I-Letrozole (i-Femara) isetshenziselwa ukwelapha umdlavuza webele kwabesifazane be-postmenopausal.I-Letrozole ivame ukunikezwa abesifazane abaye bathatha i-tamoxifen (Nolvadex, Soltamox) iminyaka engu-5.I-Letrozole iyi-non-steroidal aromatase inhibitor (yehlisa ukukhiqizwa kwe-estrogen).
I-Letrozole itholakala ngefomu elejwayelekile.Imiphumela emibi evamile ihlanganisa ukushisa okushisayo, ukuqothuka kwezinwele, ubuhlungu bamalunga/amathambo/imisipha, ukukhathala, ukujuluka okungavamile, isicanucanu, isifo sohudo, isiyezi, kanye nenkinga yokulala.
Umthamo onconyiwe we-Letrozole yithebhulethi eyodwa ye-2.5 mg elawulwa kanye ngosuku, ngaphandle kokubheka ukudla.
Ezinye izidakamizwa zingase zihlanganyele ne-Letrozole.Tshela udokotela wakho yonke imithi kadokotela kanye ne-over-the-counter kanye nezithako ozisebenzisayo.I-Letrozole akufanele isetshenziswe ngesikhathi sokukhulelwa.I-Letrozole ingase ilimaze umbungu.
I-Letrozole isetshenziswa ikakhulukazi kwabesifazane ngemva kokunqamuka kokuya esikhathini.Uma usanda kunqamuka ukuya esikhathini, xoxa nodokotela wakho ngokulawula inzalo.Ungasebenzisi isilawuli sokuzalwa esiqukethe i-estrogen.Akwaziwa uma i-Letrozole idlula obisini lwebele futhi ingase ilimaze usana oluncelisayo.Ukuncelisa ibele ngenkathi usebenzisa i-Letrozole akunconywa.
Isilinganiso se-Letrozole/Femara somdlavuza webele
1:Umthamo Ojwayelekile Wabantu Abadala Womdlavuza Webele:
Ukuze isetshenziswe njengokwelashwa komugqa wokuqala kwabesifazane abangemva kokuya esikhathini abane-hormone receptor positive noma i-hormone receptor engaziwa endaweni yomdlavuza webele othuthukile noma we-metastatic.I-Femara iphinde ikhonjiswe ekwelapheni umdlavuza webele othuthukisiwe kwabesifazane abangemva kokuya esikhathini sokuqhubeka kwesifo kulandela ukwelashwa kwe-antiestrogen: ithebhulethi engu-2.5 mg ilawulwa ngomlomo kanye ngosuku ngaphandle kokubheka ukudla.
Ezigulini ezinesifo esithuthukisiwe, ukwelashwa kwe-Letrozole kufanele kuqhubeke kuze kube yilapho kubonakala ukukhula kwesimila.
2:Umthamo Ojwayelekile Wabantu Abadala Womdlavuza Webele - I-Adjuvant:
Ukuze isetshenziswe njengokwelashwa okungeziwe kwe-adjuvant yomdlavuza webele wangaphambi kwesikhathi kwabesifazane be-postmenopausal abathole iminyaka engu-5 yokwelashwa kwe-adjuvant tamoxifen: ithebhulethi engu-2.5 mg ilawulwa ngomlomo kanye ngosuku ngaphandle kokubheka ukudla.
Ubude besikhathi esifanele sokwelashwa nge-Femara akwaziwa.Ukwelashwa kufanele kuyekwe uma kukhona ukubuya kwesimila.
Anti-Estrogens Series Product
Uchungechunge lwe-Anti-estrogen | |
I-Tamoxifen Citrate | Inombolo ye-CAS: 563.64 |
I-Clomifene Citrate | Inombolo ye-CAS: 50-41-9 |
I-Toremifene Citrate | Inombolo ye-CAS: 89778-27-8 |
I-Exemestane | Inombolo ye-CAS: 107868-30-4 |
I-Anastrozole | Inombolo ye-CAS: 120511-73-1 |
I-Letrozole | Inombolo ye-CAS: 112809-51-5 |
I-Fulvestrant | Inombolo ye-CAS: 129453-61-8 |